Teacher’s Profile
1.
Personal Details
Name
Uday Vinayakrao Desai
Designation
Professor in Organic Chemistry
Date of Birth
5th December 1956
E-mail Address
[email protected];
[email protected]
Permanent Address
Swanand, 21, Shirgaonkar Housing
Society, Rajarampuri, 8th Lane, Takala,
KOLHAPUR – 416008.
2.
3.
Academic Details:
Qualification
M. Sc.; Ph. D.
Specialization
Organic Chemistry
Position
Professor in Organic Chemistry
Research specialization
Synthetic Organic Chemistry:
Studies in the development of green
synthetic methodologies and terpenoids
Total
: 26 years
1
Teaching experience:
Page
4.
5.
U. G.
: 6 years
P. G.
: 20 years
Research Guidance
P.G. Programs:
M.Sc. Projects : 25
M. Phil. : 02
Ph. D. (Declared) : 07
Ph. D. (Working) : 06
6.
Research Publications
National : 07
International : 37
7.
Conferences Attended
National : 8
International : 1
Invited Talk : 2
Research Projects
a)
Studies in the
development of new
synthetic
methodologies
b)
Funding
Agency
Period
Grant
sanctioned/
Amount
mobilized
in Rs.
Status
UGC,
1st January
2005 – 31st
December
2007
6,91,000/-
Completed
1st April 2009
– 31st arch
2012
9,76,800/-
New Delhi
Studies in the
UGC,
Development of
Green
New Delhi
synthetic
Methodologies
successfully
Completed
successfully
2
Title of the project
Page
8.
9.
Membership/Other Charges
NIL
10.
Honors /Rewards
(a) Summer research fellow
of Indian Academy of
Sciences, 2004
(b) Worked as INSA visiting
fellow, 2008
11.
List of Publications
Pl. see annexure - I
12.
List of Conference/Workshop
/ Seminar attended
Pl. see annexure - II
Annexure – I
(LIST OF PUBLICATIONS)
1
Nickel ferrite nanoparticles - hydrogen peroxide: A green catalyst - oxidant
combination in chemoselective oxidation of thiols to disulfides and sulphides
to sulfoxides
Aparna M. Kulkarni,a Uday V. Desai,*a Kapil S. Pandit,a Makarand A.
Kulkarni,a Prakash P. Wadgaonkarb
RSC advances 2014 (in press)
2
Smple, economical, and environmentally benign protocol for the synthesis of
2-amino 3,5 - dicarbonitrile-6-sulfanyl pyridines at ambient temperature
Uday V. Desai*, Makarand A. Kulkarni, Kapil S. Pandit, Aparna M. Kulkarni
and Prakash P. Wadgaonkar
Green Chemistry Letters and Reviews, 2014,
http://dx.doi.org/10.1080/17518253.2014.925144
3DQSAR, Pharmacophore identification studies on series of indole derivatives
as dopamine antagonists
Pharmacophore 2012, 3(5), 280 -28.
3
S. D. Metkar; M. S. Bhatia; U. V. Desai
Page
3
4
Synthesis and biological evaluation of novel azetidine derivatives as
dopamine antagonist
S. D. Metkar; M. S. Bhatia; U. V. Desai
Medicinal
5
Chemistry Research (2013) 22:5982–598.
Diethylamine: A smart organocatalyst in eco-safe and diastereoselective
synthesis of medicinally privileged 2-amino-4H-chromenes at ambient
temperature
M. A. Kulkarni a, K.S. Pandi, U.V. Desai *, U. P. Lad, P. P. Wadgaonkar
Comptes Ren. Chimie, 2013, 16 (6), 689 - 695.
6
Mechanistic approach for expeditious and solvent-free synthesis of
a-hydroxy phosphonates using potassium phosphate as catalyst
M. A. Kulkarni, U. P. Lad, U. V. Desai *, S. D. Mitragotri, P. P. Wadgaonkar
Comptes Ren. Chimie, 2013, 16 (1), 148 -152.
7
A practical and highly efficient protocol for multicomponent synthesis of bphosphonomalononitriles and 2-amino-4H-chromen-4-yl phosphonates using
diethylamine as a novel organocatalyst.
M.A. Kulkarni, V.R. Pandurangi, U.V. Desai , P.P. Wadgaonkar
Comptes Ren. Chimie, 2012, 15 (12), 745- 752.
8
Potassium phosphate catalyzed efficient synthesis of 3- carboxycoumarins.
Kedar A Undale, Dipak S Gaikwad, Tarannum S Shaikh, Uday V Desai,
Dattaprasad M Pore.
Indian Journal of Chemistry, 2012, 51 B, pp. 1039-1042
9
Lithium tetrafluoroborate catalyzed highly efficient inter- and intramolecular
aza-Michael addition with aromatic amines.
Lad, U.P.; Kulkarni, M.A.; Desai, U.V.; Wadgaonkar, P.P.
Comptes Ren.Chimie, 2011, 14 (12), 1059-1064.
Silica supported orthophosphoric acid (H3PO4. SiO2): A green, heterogeneous
catalyst for solvent-free oxathioacetalization of aldehydes
Green Chemistry Letters and Reviews, 2011, 4 (3), pp. 235-240.
4
Sawant, A.D., Raut, D.G., Deorukhkar, A.R., Desai, U.V., Salunkhe, M.M.
Page
10
11
An ester appending multifunctional ionic liquid for Pd(II) catalyzed Heck
reaction.
Sawant, A.D., Raut, D.G., Darvatkar, N.B., Desai, U.V., Salunkhe, M.M.
Catalysis Communications, 2010, 12 (4), pp. 273-276.
12
Envirocat EPZ-10: A solid acid catalyst for the synthesis of 1,8-dioxooctahydro-xanthenes in aqueous medium.
Pore, D.M., Shaikh, T.S., Patil, N.G., Dongare, S.B., Desai, U.V.
Synthetic Communications, 2010, 40 (15), pp. 2215-2219.
13
Potassium phosphate catalyzed a rapid three-component synthesis of
tetrahydrobenzo[b] pyran at ambient temperature.
Pore, D.M., Undale, K.A., Dongare, B.B., Desai, U.V.
Catalysis Letters, 2009, 132 (1-2), pp. 104-108.
14
Sulfamic acid: An efficient and cost-effective solid acid catalyst for the
synthesis of a-aminophosphonates at ambient temperature.
Mitragotri, S.D., Pore, D.M., Desai, U.V., Wadgaonkar, P.P.
Catalysis Communications, (2008) 9 (9), pp. 1822-1826.
15
Trichloroisocyanuric acid-mediated one-pot synthesis of unsymmetrical 2,5disubstituted 1,3,4-oxadiazoles at ambient temperature.
Pore, D.M., Mahadik, S.M., Desai, U.V.
Synthetic Communications, 2008, 38 (18), pp. 3121-3128.
16
Lithium tetrafluoroborate-catalyzed solventless synthesis of α-aminonitriles.
Desai, U.V., Mitragotri, S.D., Thopate, T.S., Pore, D.M., Wadgaonkar, P.P.
Monatsh fur Chemie, 2007, 138 (8), pp. 759-762.
17
Anhydrous magnesium sulfate mediated solvent-free synthesis of dihydropyrimidin-2(1H)-ones at ambient temperature.
Pore, D.M., Desai, U.V., Thopate, T.S., Wadgaonkar, P.P.
Australian Journal of Chemistry, 2007, 60 (6), pp. 435-438.
Efficient synthesis of chalcones at room temperature in the presence of
Pore, D.M., Desai, U.V., Thopate, T.S., Wadgaonkar, P.P.
5
potassium phosphate.
Page
18
Russian Journal of Organic Chemistry, 2007, 43 (7), pp. 1088-1089.
19
Potassium phosphate or silicasulfuric acid catalyzed conjugate addition of
thiols to a,b- unsaturated ketones at room temperature under solvent-free
conditions.
Pore, D.M., Soudagar, M.S., Desai, U.V., Thopate, T.S., Wadagaonkar, P.P.
Tetrahedron Letters, 2006, 47 (52), pp. 9325-9328.
20
An efficient deprotection of dithioacetals to carbonyls using Oxone-KBr in
aqueous acetonitrile.
Desai, U.V., Pore, D.M., Tamhankar, B.V., Jadhav, S.A., Wadgaonkar, P.P.
Tetrahedron Letters, 2006, 47 (48), pp. 8559-8561.
21
An efficient, solvent-free method for the chemoselective synthesis of acylals
from aldehydes and their deprotection catalyzed by silica sulfuric acid as a
reusable solid acid catalyst.
Desai, U.V., Thopate, T.S., Pore, D.M.,
Wadgaonkar, P.P.
Catalysis Communications, 2006, 7 (7), pp. 508-511.
22
A Highly Efficient Synthesis of trisubstituted Quinolines using Sodium
Hydrogen sulfate on Silica-Gel as a reusable Catalyst.
U. V. Desai; S. D. Mitragotri; T. S. Thopate; D. M. Pore; P. P. Wadgaonkar
ARKIVOC, 2006, xv, 198 - 204.
23
A mild, expedient, solventless synthesis of bis (indolyl) alkanes using silica
sulfuric acid as a reusable catalyst.
Pore, D. M., Desai, U. V., Thopate, T. S., Wadgaonkar, P. P.
ARKIVOC, 2006 (12), pp. 75-80.
24
Chemoselective dithioacetalization of aldehydes using silica sulfuric acid as a
reusable catalyst.
Pore, D.M., Desai, U.V., Mane, R.B., Wadgaonkar, P.P.
Indian Journal of Chemistry - B Organic and Medicinal Chemistry,
2006 45 (5), pp. 1291-1295.
glycol)-400 as a phase transfer catalyst.
Shedge, A.S., Kavitake, B.P., Desai, U.V., Wadgaonkar, P.P.
6
A simple method for synthesis of methylene dioximes using poly(ethylene
Page
25
Synthetic Communications, 2004, 34 (24), pp. 4483-4486.
26
Comparative study of Heck reaction under thermal and microwave conditions.
Solabannavar, S.B., Desai, U.V., Mane, R.B.
Indian J. of Chem.- B Org. and Medicinal Chemistry,
2004, 43 (10), pp. 2235-2237.
27
Chemoselective tetrahydropyranylation of alcohols and their
detetrahydropyran-ylation using silicasulphuric acid as a reusable catalyst.
Pore, D.M., Desai, U.V., Mane, R.B., Wadgaonkar, P.P.
Synthetic Communications, 2004, 34 (12), pp. 2135-2142.
28
One Pot Synthesis of Monoalkylated and Mixed, Dialkylated Meldrum's Acid
Derivatives.
Desai, U.V., Pore, D.M., Mane, R.B., Solabannavar, S.B., Wadgaonkar, P.P.
Synthetic Communications, 2004, 34 (1), pp. 25-32.
29
Potassium Phosphate Catalyzed Nitroaldol Reaction.
Desai, U.V., Pore, D.M., Mane, R.B., Solabannavar, S.B., Wadgaonkar, P.P.
Synthetic Communications, 2004, 34 (1), pp. 34-39.
30
A novel short synthesis of norbisabolide.
Solabannavar, S.B., Wadgaonkar, P.P., Desai, U.V., Mane, R.B.
Indian J. of Chem. B Organic and Medicinal Chemistry, 2004,
43 (1), pp. 189-191.
31
A short synthesis of ar-todomatuic acid and dihydro-ar-turmerone by the
heck reaction.
Solabannavar, S.B., Wadgaonkar, P.P., Desai, U.V., Mane, R.B.
Organic Preparations and Procedure International, 2003,
35 (4), pp. 418-420.
32
Microwave assisted hydrolysis of Meldrum's acid derivatives and decarboxylation of derived malonic acids.
Helavi, V.B., Solabannavar, S.B., Desai, U.V., Mane, R.B.
Application of amberlite IRA-400 (basic) as a base in heck reaction.
Page
33
7
Journal of Chemical Research (S), 2003, 3, pp. 174-175.
Solabannavar, S.B., Helavi, V.B., Desai, U.V., Mane, R.B.
Synthetic Communications, 2003) 33 (3), pp. 361-365.
34
Heck reaction in aqueous medium using Amberlite IRA-400 (basic).
Solabannavar, S.B., Desai, U.V., Mane, R.B.
Green Chemistry, 2002, 4 (4), pp. 347-348.
35
A novel short synthesis of norbisabolide.
Solabannavar, S.B., Helavi, V.B., Desai, U.V., Mane, R.B.
Tetrahedron Letters, 2002, 43 (25), pp. 4535-4536.
36
Oxidation of alkylcyanohydrazines to azo-bis nitriles using Oxone-potassium
bromide in aqueous medium.
Tamhankar, B.V., Desai, U.V., Mane, R.B., Kulkarni, P.P., Wadgaonkar, P.P.
Synthetic Communications, 2002, 32 (23), pp. 3643-3646.
37
A simple and practical halogenation of activated arenes using potassium
halide and oxone® in water-acetonitrile medium.
Tamhankar, B.V., Desai, U.V., Mane, R.B., Wadgaonkar, P.P., Bedekar, A.V.
Synthetic Communications, 2001, 31 (13), pp. 2021-2027.
38
Deuterium labelling studies with aliphatic amines.
Desai, U.V., Kadam, A.J., Mane, R.B.
Indian J. of Chem-Sect- B Organic and Medicinal Chemistry, 2000,
39 (12), pp. 961-962.
39.
Synthesis of (±)-7,8- and 5,6-dimethyl-2-(2-hydroxyisopropyl) tetralins.
Desai, U.V., Kadam, A.J., Mane, R.B.
Indian J. of Chem-Sect- B Org. and Medicinal Chemistry, 2000,
39 (10), pp. 752-756.
40.
A simple and efficient oxidation of hydrazides to N,N’-diacylhydrazines using
Oxone® in an aqueous medium.
Kulkarni, P.P., Kadam, A.J., Desai, U.V., Mane, R.B., Wadgaonkar, P.P.
Journal of Chemical Research (S), 2000, 4, pp. 184-185.
free conditions under microwave irradiation.
8
Demethylation of methyl aryl ethers using pyridine hydrochloride in solvent-
Page
41.
Kulkarni, P.P., Kadam, A.J., Mane, R.B., Desai, U.V., Wadgaonkar, P.P.
Journal of Chemical Research (S), 1999, 6, pp. 394-395.
42.
Synthesis of deuterium labelled acids.
Kadam, A.J., Desai, U.V., Mane, R.B.
Journal of Labelled Compounds and Radiopharmaceuticals,
1999, 42 (9), pp. 835-842.
43.
Synthesis of 1,2-dimethyl-6-(2′-hydroxy-isopropyl)-7-methoxynaphthalene,
an isomer of emmotin-G methyl ether.
Bachute, M. T., Desai, U.V.,Mane, R.B
Indian Journal of Chemistry Section-B Organic and Medicinal
Chemistry, 1998, 37 (9), pp. 857-860.
Efficient Approach for 4-benzyl-5, 5-dimethyldihydrofuranones: Total
Synthesis of (+/-) solafuranone.
Srikrishna, A.; Satyanarayana, G.; Desai, U. V.
9
Synthetic Communications, 2007, 37 (6), 965- 976.
Page
44