Top 200 Pharmaceutical Products by US Retail Sales in 2011 Compiled and Produced by the Njardarson Group (The University of Arizona): Edon Vitaku, Elizabeth A. Ilardi, Jón T. Njarðarson Lipitor 1 (Atorvastatin) $7,688 Million CHOLEST&TRIGLY.REGULATOR 21 Avastin (Bevacizumab) Plavix 2 (Clopidogrel) Vyvanse (Lisdexamfetamine) PSYCHOSTIMULANTS 61 Humalog (Insulin Lispro) Atripla 22(Tenofovir & Emtricitabine & Efavirenz) HIV ANTIVIRALS 42 Suboxone (Buprenorphine & Naloxone) 62 Adderall XR (Amphetamine & Dextroamphetamine) (Methylphenidate) PSYCHOSTIMULANTS 101 Cubicin (Daptomycin) ANTIBACTERIAL 121 Humalog KwikPen (Insulin Lispro) HUMAN INSULIN+ANALOGUES 141 Forteo (Teriparatide) PARATHYROID HORM&ANALOGS 161 Xifaxan (Rifaximin) ANTIBACTERIAL 181 Yervoy (Ipilimumab) ANTICANCER HandiHaler 23 Spiriva (Tiotropium Bromide) Synagis (Palivizumab) SPEOF. IMM-GLOB. ANTIVIRAL 102 Boniva (Ibandronate) BONE CALCIUM REGULATORS 122 Pegasys Conv. Pack (Peginterferon Alfa-2a) ANTIVIRALS EXCL ANTI-HIV 142 Avapro (Irbesartan) 43 (Atorvastatin) 63 Exforge (Amlodipine & Valsartan) ANGIOTEN-II ANTAG, COMB Reference http://www.pharmacytimes.com/publications/issue/2012/July2012/Top-200-Drugs-of-2011 (Lidocaine) Neupogen (Filgrastim) 83 Venlafaxine HCl ER (Venlafaxine) ANTIDEPRESS.& MOOD STAB. LAR 103 Sandostatin (Octreotide Acetate) HYPOTHALAMIC HORMONES 123 Gammagard Liquid (Immune Globulin) IMMUNOMODULATORY AGENTS 143 Mirena (Levonorgestrel) CONTRACEPTIVES 163 NovoSeven RT (Eptacog Alpha) 24 Januvia (Sitagliptin) DPP-IV INHIBITOR A-DIABS 44 Onglyza (Saxagliptin) ANTIDIABETIC Procrit (Epoetin Alfa) ERYTHROPOIETIN PRODUCTS 64 (Fluticasone & Salmeterol) Flovent HFA (Fluticasone Propionate) 84 Restasis (Cyclosporine) IMMUNOSUPPRESSIVE AGENTS 104 Actonel (Risedronate) BONE CALCIUM REGULATORS 124 Prograf (Tacrolimus) 25 Lantus (Insulin Glargine) TYPE 2 DIABETES PRODUCT 164 Bystolic (Nebivolol) B-BLOCKING AGENTS 184 Abraxane (Paclitaxel) ANTICANCER (Quetiapine) $4,637 Million ANTIPSYCHOTICS 26 Truvada (Tenofovir & Emtricitabine) HUMAN INSULIN+ANALOGUES 45 Eloxatin (Oxaliplatin) ALL OTH. ANTINEOPLASTICS 65 ProAir HFA (Salbutamol) 85 Zyvox (Linezolid) 46 Niaspan (Niacin) Sensipar (Cinacalcet) 66 Reyataz (Atazanavir) Treanda (Bendamustine) 86 Betaseron (Interferon Beta-1b) Zosyn (Pipperacillin & Tazobactam) ENZYME INHIBITORS 165 Invega Sustenna (Paliperidone palmitate) ANTIPSYCHOTIC Hydrocodone/APAP 185(Hydrocodone & Acetaminophen) ANALGESICS 27 Diovan (Valsartan) 47 Provigil PSYCHOSTIMULANTS 67 Aciphex (Rabeprazole) 126 Risperdal Consta (Risperidone) 87 Evista (Raloxifene) Exelon (Rivastigmine) ANTI-ALZHEIMER PRODUCTS 166 Lialda (Mesalazine) INTESTINAL ANTIINFLAMM 186 Synvisc-One (Hylan G-F 20) OSTEOARTHRITIS $4,404 Million CHOLEST&TRIGLY.REGULATOR 28 Asacol (Mesalazine) INTESTINAL ANTIINFLAMM 127 Colcrys (Colchicine) 48 Privigen (Human Immune Globulin) IMMUNOMODULATORY AGENTS 167 Gilenya (Fingolimod) MULTIPLE SCLEROSIS Zydis 187 Zyprexa (Olanzapine) ANTIPSYCHOTICS Aranesp (Darbepoetin alfa) ERYTHROPOIETIN PRODUCTS 68 Concerta (Methylphenidate) PSYCHOSTIMULANTS 88 Erbitux (Cetuximab) ANTICANCER Loestrin 24 Fe 108 (Norethindrone Acetate & Ethynyl Estradiol) HORMONAL CONTRACEPT SYST 128 ANTIARTHRITIS 147 Lyrica (Pregabalin) ANTIEPILEPTICS SERMS ANTIPSYCHOTICS 146 (Rosuvastatin) ANTIULCERANTS Amphetamine Salts ER 107 106 (Amphetamine & Dextroamphetamine) PSYCHOSTIMULANTS Crestor 8 ANGIOTEN-II ANTAG, PLAIN INTERFERONS ANTICANCER 145 $4,593 Million ANTILEUK ANTIASTHMATICS HIV ANTIVIRALS PARATHYROID HORM.REGULATOR 125 (Montelukast) CHOLEST&TRIGLY.REGULATOR OTHER ANTIBACTERIALS 105 Singulair 7 HIV ANTIVIRALS B2-STIMULANTS IMMUNOSUPPRESSIVE AGENTS 3-Pak 144 Victoza (Liraglutide) Seroquel 6 $4,637 Million CORTICOIDS CORTICOIDS BLOOD COAGULATION 183 Advair Diskus 5 $5,194 Million ANTIPSYCHOTICS CORTICOIDS CHOLEST&TRIGLY.REGULATOR 182 Lidoderm ANAESTHETICS, LOCAL ANGIOTEN-II ANTAG, PLAIN 162 Atorvastatin Calcium (Aripiprazole) CHR. OBS. PULMONARY DIS. PSYCHOSTIMULANTS 82 Abilify 4 $6,156 Million ANTIULCERANTS DRUGS USED IN OPIOID DEP HUMAN INSULIN+ANALOGUES 81 Methylphenidate ER (Esomeprazole) $6,711 Million PLATELET AGGR.INHIBITORS ALL OTH. ANTINEOPLASTICS 41 Nexium 3 Norvir (Ritonavir) HIV ANTIVIRAL 148 Revlimid (Lenalidomide) IMMUNOSUPPRESIVE AGENTS 168 Pneumovax 23 (Pneumococcal Polyvalent) PURE VACCINES HCl XL 188 Bupropion (Bupropion) ANTIDEPRESSANT Cymbalta 9 (Duloxetine) $3,666 Million ANTIDEPRESS.& MOOD STAB. 29 Celebrex (Celecoxib) Humira 10 (Adalimumab) $3,531 Million SPEC ANTIRHEUMATIC AGENT 30 Lucentis (Ranibizumab) ANTIRHEUMATIC N-STEROID 49 Androgel (Testosterone) ANDROGENS, EXCL G3E,G3F 69 Budesonide (Budesonide) IMMUNOSTIM. AG. EX. INTFRON. 89 Benicar (Olmesartan) ANGIOTEN-II ANTAG, PLAIN 109 Tarceva (Erlotinib) ANTIANGIOGENICS 50 Combivent (Ipratropium & Salbutamol) 70 Levemir (Insulin Detemir) Premarin (Conjugated Estrogens) OESTROG EX G3A,G3E,G3F 149 Lexiscan (Regadenoson) Velcade (Bortezomib) ALL OTH. ANTINEOPLASTICS Pradaxa 110 (Dabigatran) ANTICOAGULANT 130 Effexor XR (Venlafaxine) ANTIDEPRESS.& MOOD STAB. 189 Qvar (Beclometasone Dipropionate) GLUCOCORTICOID Nuvaring (Etonogestrel & Ethynyl Estradiol) 150 Stelara (Ustekinumab) 51 Kaletra (Lopinavir & Ritonavir) 71 32 Lovenox (Enoxaparin) Diovan HCT (Valsartan & Hydrochlorothiazide) Incivek (Telaprevir) 91 Zometa (Zoledronic Acid) 52 Rebif (Interferon Beta-1a) Renvela (Sevelamer) HYPERKAL.HYPERPHOS.PRODS 131 Xopenex (Salbutamol) B2-STIMULANTS 72 Varivax (Varicella Zoster) 171 Flexpen Mix 191 190 NovoLog (Insulin Aspart) Zostavax (Herpes Zoster) PURE VACCINES Maxalt MLT (Rizatriptan) ANTIMIGRAINE PREPS 33 Avonex (Interferon Beta-1a) INTERFERONS 53 Vytorin (Simvastatin & Ezetimibe) 92 Synthroid (Levothyroxine) ANTIARTHRITIC 112 Gamunex-C (Human Immune Globulin) IMMUNOMODULATORY AGENTS 132 Travatan Z (Travoprost) 73 172Metoprolol Succinate (Metoprolol Succinate) Zemplar (Paricalcitol) VIT. A & D INC. COMBS. $3,316 Million IMMUNOSTIM AG. EX. INTFRON. SoloSTAR 34 Lantus (Insulin Glargine) HUMAN INSULIN+ANALOGUES 54 Nasonex (Mometasone) TOPICAL NASAL PREPS 74 ANTIBACTERIAL 93 Vesicare (Solifenacin) Lunesta (Eszopiclone) HYPNOTICS & SEDATIVES 94 URINARY INCONTINENCE PRD 113 Pristiq (Desvenlafaxine) 133 Epzicom (Lamivudine & Abacavir) 114 Welchol (Colesevelam) 134 Taxotere (Docetaxel) 154 Docetaxel (Docetaxel) VINCA ALKALOIDS Angiomax (Bivalirudin) 174 Tysabri (Natalizumab) 35 Vancocin (Vancomycin) ANTIBIOTIC (Rituximab) Zyprexa 16 (Olanzapine) Gleevec (Imatinib) $2,965 Million ANTIPSYCHOTICS 36 Namenda (Memantine) ALL OTH. ANTINEOPLASTICS 55 Viagra ERECTILE DYSFUNCTION PRD 75 Cialis ANTIALZHEIMER 56 Symbicort (Budesonide & Formoterol) 95 Detrol LA (Tolterodine) URINARY INCONTINENCE PRD 115 Trilipix 76 Solodyn (Minocycline) ANTIBIOTIC 96 Opana ER (Oxymorphone) DRUGS USED IN OPIOID DEP Focalin XR 116 (Dexmethylphenidate) CHOLEST&TRIGLY.REGULATOR (Amphetamine & Dextroamphetamine) Gardasil 155(Human Papillomavirus Quadrivalent) PURE VACCINES 175 Donepezil HCl (Donepezil) ANTI-ALZHEIMER 195 Lamictal (Lamotrigine) ANTIEPILEPTICS (Glatiramer Acetate) $2,956 Million IMMUNOSTIM AG EX INTFRON Sodium 37 Enoxaparin (Enoxaparin) Fentanyl (Fentanyl) 57 Seroquel XR (Quetiapine) Lumigan (Bimatoprost) 77 NovoLog FlexPen (Insulin Aspart) Chantix (Varenicline) 97 Orencia (Abatacept) Menactra (Meningococcal Conjugate) ANTIMENINGITIS Geodon (Ziprasidone) ANTIPSYCHOTICS 58 Alimta (Pemetrexed) ANTIMETABOLITES 78 Isentress (Raltegravir) 117 Avodart (Dutasteride) BPH PRODUCTS 137 Actoplus Met (Metformin & Pioglitazone) ANTIDIABETIC 157 Pulmozyme (Dornase Alfa) 98 Prezista (Darunavir) Xgeva (Denosumab) OSTEOPOROSIS 197 Vidaza (Azacitidine) ANTICANCER $2,880 Million NARCOTIC ANALGESICS 39 Zetia (Ezetimibe) CHOLEST&TRIGLY.REGULATOR 59 Novolog (Insulin Aspart) HUMAN INSULIN+ANALOGUES 79 Levaquin FLUORO-QUINOLONES 99 Ventolin HFA (Salbutamol) HIV ANTIVIRALS Xolair 118 (Omalizumab) ALL OTH. A-ASTHMA & COPD. 138 Aggrenox (Dipyridamole & Aspirin) B2-STIMULANTS Strattera 119 (Atomoxetine) ALL OTHER CNS DRUGS 139 PLATELET AGGR.INHIBITORS 158 CYSTIC FIBROSIS 177 (Oxycodone) HIV ANTIVIRALS ANTIRHEUMATIC AGENTS ANTISMOKING PRODUCTS 196 38 Oxycontin 19 $2,926 Million ANTIDEPRESS.& MOOD STAB. HUMAN INSULIN+ANALOGUES MIOTICS+ANTIGLAUC.PREPS 176 (Escitalopram) ANTIPSYCHOTICS NARCOTIC ANALGESICS 156 Lexapro 18 HUMAN INSULIN+ANALOGUES PSYCHOSTIMULANTS 135 Amphetamine Salts ER 136 PSYCHOSTIMULANTS Copaxone 17 B2-STIMULANTS+CORTICOIDS ERECTILE DYSFUNCTION PRD MULTIPLE SCLEROSIS 194 Rituxan $3,005 Million ALL OTH. ANTINEOPLASTICS ANTITHROMBOTIC ANTICANCER 193 Aloxi (Palonosetron) 15 ANTIEMETIC CHOLEST&TRIGLY.REGULATOR 173 Dexilant (Dexlansoprazole) ANTIULCERANTS HIV ANTIVIRALS 153 Xeloda (Capecitabine) ANTIMETABOLITES ANTIDEPRESS.& MOOD STAB. ANTIARRHYTHMIC AGENTS 192 Prevnar 13 (Pneumococcal 13-Valent Conjugate) MIOTICS+ANTIGLAUC.PREPS. HORMONAL CONTRACEPT SYST Neulasta 14 LIP.REG.CO.W.OTH.LIP.REG PURE VACCINES Adacel Ortho Tri Cyclen Lo 151 152(Norgestimate (Ttns. Tox. & Rdcd. Diphth. Tox. & Acel. Pert.) & Ethynyl Estradiol) VACCINES $3,438 Million GLITAZONE ANTIDIABETICS INTERFERONS BONE CALCIUM REGULATORS 111 (Pioglitazone) ANGIOTEN-II ANTAG, COMB ANTIVIRAL HIV ANTIVIRALS HUMAN INSULIN+ANALOGUES (Trastuzumab) Actos 13 $3,474 Million IMMUNOSUPPRESSIVE AGENTS HEPARINS ANTIPSORIASIS 170 Herceptin Remicade 12 ALL OTH. ANTINEOPLASTICS HORMONAL CONTRACEPT SYST CORONARY VASODILATOR 169 31 HUMAN INSULIN+ANALOGUES 90 Enbrel (Etanercept) $3,507 Million SPEC ANTIRHEUMATIC AGENT ANTICHOLINERGIC+B2-STIM ALL OTH. ANTINEOPLASTICS 129 11 Invega (Paliperidone) Nutropin AQ (Somatropin) 159 Valcyte (Valganciclovir) HIV AND CMV ANTIVIRAL Reclast (Zoledronic Acid) (Epoetin Alfa) $2,774 Million ERYTHROPOIETIN PRODUCTS 40 Tricor CHOLEST&TRIGLY.REGULATOR 60 Lovaza (Omega-3-Acid Ethyl Esters) ANTIATHEROMA NATRL ORIG 80 Janumet (Sitagliptin & Metformin) DPP-IV INHIBITOR A-DIABS 100 ANGIOTEN-II ANTAG, COMB 120 140 Metoprolol Succinate (Metoprolol Succinate) ANTIARRHYTHMIC AGENTS 160 CORTICOIDS (Iohexol) LOW OSMOLAR ANGIO-UROGRP. Temodar (Temozolomide) ALKYLATING AGENTS (Fluticasone Propionate) Omnipaque Byetta (Exenatide) GLP-1 AGONIST A-DIABS 179 Fluticasone Propionate 180 199 Benicar HCT (Olmesartan & Hydrochlorothiazide) OSTEOPOROSIS HORMONE REPLACEMENT AGENTS 198 (Tenofovir) HIV ANTIVIRALS ANTIPSYCHOTICS 178 Viread Epogen 20 Avelox FLUORO-QUINOLONES 200 Ranexa (Ranolazine) ANGIOTEN-II ANTAG, PLAIN
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