IND@COF MA.TERIAI@S This index refers to the present compilation only. A cumulative index will appear at the end of this year for all issues in this series of supp1en@nts to CANCER RPZEARcH. @teria1s found in the article, Toxicity and Antileukemic Effectiveness of Pyridine Derivatives az@ 1,3,4-Thiadiazole Derivatives in Mice Relationship to Nico tin@mide Antagonism.@p. 483—550), are tabulated by NSC Numbers, or by cc*upound name if' there is no NBC Number for the n@teria1, in the various tables of the article. To find detailed data for cctigounds listed in the index as Thitry Numbers 29946-29993, the reader should go to the Swmnary Table A (pp. 497-500), which contains a cross index contaiPin@ P2@TRYNumber, NSC Number, Compound 551 Name and Table Number. CancerResearch 552 ENTRY FORMULAS NOS' ENTRY FORMULAS NOS. FORMULAS ENTRY NOS. C6 CS C C H5 . N3 1/2 29941 0 H2 S 04 29011 C H5 04 P 29014 (2 ((2 H2 02)X (2 H3 N3 S C2 C2 C2 C2 H4 H6 H7 H7 (2 H15 CL AS 29406 29978 N6 0 03 S N 0 • HCL 04 P 0 29850 29008 28818 29012 29069 . H2 0 C3 (3 (3 H2 H4 29851 0 0 CL6 CL2 79356 ((3 H4 N2 02)X (3 H5 • (4 (3 (3 C3 (3 (3 (3 H5 H5 N H4 04 N3 N3 02 03 H5 N3 S H6 03 S H7 N3 •HBR H9 04 p 29390 29740 29904 29942 29984 29905 29656 29015 (4 H5 CL3 C4 C4 C4 (4 (4 (4 (4 H5 HS H5 HS HS H6 H6 CL4 N 02 F3 0 N 02 52 N S N3 0 S 8R4 0 N4 (4 H6 53 C4 (4 (4 C4 (4 (4 C4 H7 H7 H7 H7 H8 H8 H9 CL2 F 0 N 0 N? 03 N3 S N2 02 02 N 0 S N 02 52 (4 H9 C4 (4 (4 (4 (4 H9 N 03 H9 N 52 H10 N 05 P H10 N4 02 Hil 04 P 5 29007 29628 29447 28900 28913 29264 29186 29411 29979 29391 28848 28902 29265 29449 29906 29980 29392 28819 29719 29433 28967 28909 29428 29393 29017 29016 CS H6 N2 03 S CS H6 OS 52 CS H7 BR N2 02 H2 H3 H3 H3 H3 H3 H4 02 H4 H4 H4 HS HS HS HS HS HS BR 12 N 02 BR I N 02 8R2 N 02 CL2 N 02 CL3 12 N 02 AS CL2 AS 12 N 02 CL N 02 F N 02 AS 0 CL N2 0 I N2 02 N 0 N 02 N 03 29585 29588 . . (6 (6 (6 (6 . 29600 29182 28863 29118 29020 29987 (6 (6 (6 C6 (6 (6 (6 C6 H6 H6 H7 H7 H7 H7 H7 H7 •(7 N2 S 03 AS 04 CL N2 0 5 CL3 03 S2 N 0 N3 0 02 P H17 H9 (6 (6 (6 (6 (6 (6 C6 (6 (6 C6 C6 (6 H9 F3 0 H9 N S H10 BR2 02 H10 CL 0 P S H10 N2 02 H10 03 H10 03 S2 Hil CL2 F 0 H11 I OS Hil N 57 H12 N2 0 H13 N (6 CL2 H3 F 0 N3 CL 03 7 5 N OS P 04 P 0 512 29908 29429 29019 29543 29580 29502 28951 29060 29959 29144 29952 29412 29970 29954 28864 K 28993 29591 SALT C7 H4 CL2 0 (7 H4 CL2 02 (7 H5 AS 12 02 C7 H6 N4 OS C7 H7 CL N2 0 (7 H7 CL 02 S (7 H7 F7 0 (7 H7 N 0 (7 H7 N 02 (7 H7 N 02 S (7 HR N2 0 (7 H8 N2 0 5 C7 H8 04 (7 H8 S (7 H9 AS 03 (7 H9 AS 04 (7 H9 N 0 C7 H9 N2 02 (7 H10 BR2 02 C7 H1O 0 (7 H10 04 (7 Hil N 0 • HRR C7 H12 8R2 02 (7 H12 02 (7 H12 03 (7 H13 CL N2 0 5 28992 28995 28867 29909 29075 29000 29270 29973 29955 29189 29960 29662 29961 29533 29003 29166 29004 28868 29974 29854 29563 29657 29120 29610 29548 29271 29364 29663 29562 •HCL 29950 (7 H13 06 P (7 H13 (7 H14 C7 H14 (7 H14 (7 HiS •(4 29972 29949 CL3 N 29605 I OS N2 06 02 06 N 29451 29855 29255 29534 29107 H4 29117 04 C7 HIS rh 0 (7 H16 N OS P (7 H17 04 P 29856 29606 29452 (8 (6 . 29493 29467 N C6 H7 02 P •C18 H39 N (6 H8 N (6 H8 N2 0 S (6 H8 N4 0 (6 HR 0 (6 H9 CL 02 S 29968 29482 29488 29948 29947 29958 29660 29852 29139 29746 29590 29971 29839 29695 H14 H14 HiS H18 C7 H3 CL3 0 (7 H3 CL3 0 S2 28862 29946 29953 29162 HCL (7 29907 29018 29542 29127 29188 HCL (6 H13 N3 02 29622 28968 29990 29561 29043 29584 29181 29096 SALT C6 H6 N2 0 (6 H6 N2 02 28983 28994 28999 29658 29991 29587 29389 29266 29966 28964 29967 29969 29659 28911 29044 (6 C6 (6 (6 (6 (6 C6 N C6 (6 (6 C6 (6 C6 (6 C6 C6 • K CS CS CL2 F6 (5 CL2 F6 02 CS CL6 0 CS H4 BR N3 02 •NA SALT (5 H4 N4 S CS HS CL3 0 53 CS HS CL3 02 CS H5 FS 0 (5 H5 N C5 H6 CL N3 CS H6 N2 (6 H13 N 03 C6 H13 N S 29546 C6 (4 C4 H2 CL8 52 C4 H3 CL N2 (4 H5 CL OS CS H7 8R2 CL 02 CS H7 CL3 0 53 (5 H7 CL3 02 53 CS H7 N 02 S CS H? N3 0 CS H7 N3 04 (5 H8 8R2 02 (5 H8 N2 02 (5 H8 0 S2 CS H9 N 0 CS H10 N2 S •1/2 (4 H4 04 (5 H11 N 0 CS H11 N 0 • (6 H3 N3 07 (5 H11 04 P C5 H13 N • C6 H3 N 07 CS H13 N • HCL CS H13 N3 •1/2 (4 H4 04 CS H13 04 P CS H14 0 SI 29696 29965 29745 29956 29853 28914 29267 29268 29187 29545 29006 28820 29498 28910 29269 29450 29661 29394 28866 07 C6 H13 N 02 S 29434 (8 H4 CL2 F2 0 (8 H4 CL2 02 (8 H4 CL6 (8 HS CL F2 0 (8 HS CL N2 (8 HS CL N2 0 C8 H5 CL2 N 02 (8 H5 I 04 C8 H6 N? 02 (8 H6 N2 02 • HCL (8 H6 04 . C8 C8 (8 (8 (8 C8 (8 (8 2 H7 H7 H7 H7 HR H8 H8 H8 C8 H11 29272 28990 28988 29273 29629 29888 28963 29154 29630 29061 29062 N CL 0 CL 02 N3 02 52 N3 03 CL6 N2 02 F6 N2 02 HG N2 04 I N 02 28991 28989 28958 28962 29986 @991U 28842 29697 28871 29483 29183 Index ofMaterials FORMULASENTRYNOS.(8(8HR ENTRY FORMULAS 553 NOS. FORMULASENTRYNOS.(10(10 (9 0429505C8HR I N (9 H10 N2 02 0379957(8H8 N2 (9 H10 N2 (9 (9 C9 (9 (9 (9 (9 (9 (9 (9 (9 H10 H1O H1O H1O H1O H1O H1O Hil Hil Hil H11 N6 0 S 07 03 04 05 52 BR CL 02 CL2 04 P N 0 (9 (9 (9 (9 (9 (9 (9 Hil Hil Hil H12 H12 H12 H12 N 03 N OS NS 02 5 AS N 05 AS N 06 CL 04 p N2 0 0429843.NA N4 SALT(8HR S28839(8H8 02 5229582(8H9 04 0429664(8H9 AS CL N 0629720(8H9 AS N? 0229274C8H9 F3 29474(8H9 HG+ CL N 029275 2997529395(8H9 0429484(8H10 N3 0228841(8H10 (L4 N2 N2 029076 29416229413C8H10 N2 0229476 2996429951(8H10 0329506C8Hil 0229276(8Hil F3 N2927729278(8H11 028973.1/2 N S(8Hil H2 04 022882829737(8H12 N 0228844(8H12 RR2 N2 0228840(8H12 CL2 N2 N229279(8H12 0229036(8H12 N2 S2973629753(8H13 N2 02 029478(8H13 N 0229191(8H13 N S29190(8H13 N 028965(8H13 N3 529078(8H14 N3 02 029396(8H14 14R4 0229035(8H14 N2 029538(8H14 0.2936529631(8H14 032936629367(8HiS 0229569(8HiS CL 02976829769(8HiS N 0329124CRH16 N 0229397(8H16 N? 5229436(8H16 ‘92 04 0629134(8H16 N2 029368(8H16 022925429911CSH17 0229777.HCL(8H17 N 0329912(85118 N 029398(8H18 N2 S29009(8H19 0229735(8H19 N 04 P29021 2902379022C9(9H4 03 (9 H12 N4 02 5 (9 H12 02 (9 H13 N (9 H13 N 0 (9 H13 04 P (9 H14 N+ I— (9 H14 N2 (9 (9 (9 (9 C9 HiS H16 H16 H16 H16 N 0 bR2 02 N2 02 02 03 (9 H17 CL N2 02 • HCL (9 H17 N •HCL (9 H17 N 0 S S 29497 29038 29668 28905 29499 29229 29726 29531 28901 29683 29131 29595 29281 29369 29724 29507 29894 29725 29738 29593 29283 29414 29159 29723 29284 29286 29192 29592 29770 29287 29371 29416 29479 29547 29289 29372 29374 29113 29455 29282 29976 29594 29370 29285 29682 Hi2 0429503 29288 29415 29858 29373 0629727(10 Hi3 AS N2 H13 N 029i63 29977(10 0229918• H13 N HCL(10 S29438S H13 N 02 HCLdo HCL(10 29913 29013 29114 29228 28928 29375 29094 29914 29699 N2891502 H14 CL S(10 H14 N2 029686 29963(10 0229862(10 H14 N2 P29992(10 H14 N5 07 0429361Cio Hi4 0829457(10 Hi4 S29376Cio Hi4 N2960303 HiS CL P(10 HiS N29294 2929629295(10 N29111. HiS 04(10 (4 (10 0428982C9H4 CL6 0429665(9H6 (LB28997(9He 0229280C9H6 F3 N 5328912(9H7 0229890(9H7 N S29666(9HR N 0229667(9H8 CL3 N 0228998(9H8 CL6 5228869(9HR 0 0229857(9H8 042945429504(9H9 029501(9H9 BR 028959(9H9 CL 0228961(9H9 CL 0329535.1/2 N SALTC9H9 BA 522998529988C9H1O N3 02 0229698(9H10 CL3 N 0228977•HCL F N CL8 (L1O H5 (L2 N 0 28981 28986 2991S HS CL2 N 02 29916 H6 N2 03 52 H7 CL N 0 52 (10 H7 CL (10 do do (10 H7 H7 H7 H7 CL3 52 F3 02 N 0 52 N 0 52 29572 29573 29754 29632 29290 29574 29607 . (10 (10 (10 do (10 (10 H4 029196(10 HiS N S29197S H15 N 0 do (10 (10 52 (10 52 ClO (10 K 03 S SALT H7 H7 H8 H8 H8 H8 N 0? 52 N 03 13R4 0 CL N 02 FE N2 0 5 29575 29448 29407 29943 29859 29263 2929329292 S29456(10 H13 N3 0 0329126do H13 N3 042912129861do H13 N3 N29689S H14 CL 29360 29193 29194 28927 2977229633(10 2968529634(10 HCL (9 H17 N 02 (9 H18 CL N • HCL (9 H18 CL3 03 P (9 H18 N2 03 • (4 H4 04 (9 H18 02 (9 H19 N 0 • HCL (9 H20 N? (9 H21 N3 • (4 H4 04 (9 H21 04 p (9 H22 N2 0229565(10 H9 8R2 CL 022904529046(10 H9 CL N2 5328899(10 H9 CL 0 0229669(10 H9 CL2 N N2891602 H9 CL4 5(10 0229687• H9 N HCL(10 0529508(10 H10 PR? I-'29771(10 H1O N+ 0429684(10 H10 0829728(10 Hil AS N2 022892929532(10 Hil BR 5228906(10 H11 CL N29739(10 Hil CL4 0229291(10 Hil F7 029688(10 Hil N 032919529437(10 H11 N 028895(10 H12 CL N2 CL228996(10 H12 0329037(10 H12 N2 OLe29860(10 H12 N2 5229983do H12 N4 02 0229747(10 H12 N6 0229536do Hi? Hi2 0329500 HCLdo 29917 022882329258(10 HiS N S29895do HiS N5 02 P29601do HiS 05 CL?29743N2 H16 02do N22929729417(10 H16 H16 029786 2991929787do OS28930(10 H16 0329773do H17 N 022937729670(10 H18 0329559(10 H18 5229690(10 H18 04 $228870do H18 029198(10 H19 N 029378. H19 N HCL(10 I—28865(10 H20 N 0+ N2299402 H20 HCL 2983829837 CancerResearch 554 FORMULAS ENTRY NOS. FORMULAS FORMULASENTRY NOS.(11Cli (10 ENTRY NOS. (12 0729614CliCli (10 H20N2 528918(ii H7CL 02 H9CL 529755Cii 03 S29050Cii H9N OS 0229042(ii H1ON2 H10029729(ii H100228924(11 HilBR 0229041Cii N2 022960929671Cli N Hil(L2 528966(11 HilN3 02 022955029564(ii H128R2 0329549(ii H12BR2 OS29509Cii H128R2 0229672Cii N H12CL3 H12N22929829357Cli 029863Cli H12N2 022904029864Cli H12N2 529458(ii H12N2 02 529673(11 H12N2 08 H120 5229586Cli H120329362(ii H120429030(11 029692Cli H13N 029865• H13N HCLCli Hi3N 022969329694Cli 0329866Cli H13N 5228904Cii H13N 03 029053Cii H13N2 029717Cii N H14CL H14(L2 N2959606 PCii P29598(11 H14CL3 04 042885029867Cli Hi4N2 0529868Cii H14N2 529674(11 H14N2 06 H14N3 5+29742BR 03 . 5229002(12 H4 CL6 0429490(12 H5 8R3 N2 I28871(12 H8 AS AS228872N? H8 04(12 5229001(12 H8 CL2 N229471(12 H8 F4 5229635C12 H8 12 5229576(12 H8 N2 03 0429473(12 H8 N2 N429363(12 H8 0629145(12 H9 AS N2 0728873(12 H9 AS HiSN 0329870(11 HiSN3 0229047Cli H16I 029184(11 N Hi6N 1—28931Cii 03+ H16N229304(ii 029305Cli Hi6M2 H16N2 0229119Cii 0229844Cii H16N4 H16N4 529137Cli 02 H16029379Cli S29459Cli H1602 H17N29306 HCLCii 032940829722Cli H17N 529122Cli H17N 03 H1704 P29460Cli H18N+ 1—29112Cli H18N229310 2941829311Cli H18OS29200Cli H19NS 529160(11 02 H200329558Cli 022916429201(11 H21N 029085.HI(11 H22N2 H23N29149 . . 29829 29167 29170 29Q63 0329897(12 H10 CL NS 029312(12 H1O N2 0529899(12 H1O N6 0429636Cl? H10 N29064• Hil AS CL HCL(12 0228875(12 Hil AS 0328876(12 Hil AS 0428877(12 Hil AS 0629231(12 Hil CL 0328917(12 Hli CL4 N 0228878(12 H12 AS N 0229034(12 Hi2 N2 S228920(12 H12 N2 02 0529900(12 H12 N4 0629261(12 H12 0228879(12 H13 AS 2930229301 N2 29898 29130 29566 29638 29205 HRR H22 (4 2 N2 H4 H22 H22 H23 H23 H24 29116 04 N2 04 03 N 0 N 02 N2 29540 29700 29206 29207 29704 HCL 29256 29208 29703 29026 29026 29209 H24 03 (12 H2S N 0 (12 H26 0 H27 03 P H28 N HCL (13 29065 29202 29203 29314 29432 29701(12 OS29675(12 H15 N2 CL HCL(12 0229891(12 H16 N2 028861Ci? H16 H16 0328822 29557(12 0429637(12 H16 029702(12 Hi7 CL N29317(12 H17 0229874(12 H17 N 0328935• H17 N HCL(12 S29439Ci? H17 N3 05 H17 06 P29604 N 0 29319 29825 29539 (12 . 029889(12 HiS N 0229316(12 HiS N N29105. H16 02 04 06 29084 (12 HCLCl? N 0328934 N2 N2 N2 N2 04 S BR (12 H27 04 p N329313(12 H13 H15 H2O H20 H20 H20 H?O H2O H22 (12 H24 N2 0 .HI (12 0429168(12 H13 AS N2 529440(12 H13 N 05 028933(12 H14 N2 0229033(12 H14 N2 S29315(12 Hi4 N2 0229380(12 H14 0328852(12 H14 0428851(12 H14 0529551(12 Hi4 0329409. HiS BR N2 29318 29101 29204 29109 H19 N2 0+ 1— 29082 H19 04 p 29599 29788 H20 28845 H20 BR2 N2 Ci? (12 (12 (12 (12 . N2 N2 03 N 02 N 03 HCL (12 HCL(12 2930829307(11 02930929871Cii H17N H17N 029778. N2 0229480Cl? H9 BR N2 0228874(12 H10 AS BR I29161(12 H1O AS 0228932(12 HIM AS I 0329896(12 HlO BR P95 N29103. H10 CL H18 H18 H19 H19 (12 (12 (12 (12 02 (12 (12 (12 (12 (17 (12 (12 0429123(12 H2 N2 N22947704(12 H4 BR2 12 H14022919929691(11 (ii H140328897Cli H140429869Cii 5228907(11 HiSCL P29597Cii HiS(L2 04 H15N29299(ii 029300 H15N 29303Cii Cl? (12 (12 (12 029756Cli H24 5229783Cli H24 03 N329108.Cl?(12 H?5 29872 28860 29873 (13 (13 (13 (13 (13 (13 (13 (13 H8 (L2 0 S H8 N2 0 H9 AS BR2 0 H9 BR 02 H9 CL3 02 5 H9 N 02 H9 N 04 5 H1O BR N 03 (13 H1O CL (13 (13 C13 (13 (13 (13 C13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 (13 H10 H10 Hil Hil Hil Hil Hil Hil H12 H12 H12 H13 H13 H13 Hi4 H14 H14 HiS H16 H16 H16 H16 H16 H17 H17 H17 H17 H18 Hi8 H18 H18 N2 02 04 AS 8R2 AS 02 N N 0 N 04 N 06 N2 0 N4 02 03 N N 0 N5 04 N2 0 06 N3 0 N2 N2 0 0 02 03 N N 02 N 04 S N3 03 52 N2 •HCL N2 03 P12 04 0 N 28919 29830 29175 29210 28925 29621 29639 29640 29513 29320 29774 28936 28880 28837 29321 29461 29443 29322 29849 29641 29323 29324 29325 29901 29326 29148 29327 29328 29230 29938 29552 29329 29832 28853 29608 29705 29381 29419 29920 29444 29981 28937 29875 29420 29382 29982 Index ofMaterials FORMULAS ENTRY NOS. C13 H19 N 0 C13 H19 N 0 02 . (14 H26 N2 04 (14 H27 BR 02 (14 H30 0 29555 29744 29462 29330 29179 •2 HCL 2 H2 H22 0 N2 29331 02 29827 29945 29383 29567 C13 H24 N2 011 Cia H24 02 C13 H2S CL 02 (14 H7 H9 H9 H9 H10 N3 02 CL3 F2 N 02 N3 06 N4 06 0 C14 H1O 02 S C14 C14 H1O H1O 04 06 C14 Hil CL F2 0 C14 Hil CL 0 C14 Hil F3 0 (14 Hil N Ci4 Hil N 02 C14 Hil N 03 29831 29332 29642 29517 29399 29005 29211 29185 29333 28960 29334 29518 29335 C14 H13 AS 03 (14 H13 8R2 CL 29707 29468 28882 29494 29512 29757 29143 29466 N2 C14 29336 C14 H12 9R2 N2 C14 H12 N2 0 C14 H12 N2 04 CiA H12 0 C14 H12 H13 03 N 0 29400 29624 29921 29337 29384 C14 H13 N 04 S C14 (14 C14 C14 C14 C14 H14 H14 H14 H15 H15 H16 8R2 29625 29489 N2 29492 29487 N2 0 N2 02 N 0 N3 0 N2 H16 H16 P42 02 N2 04 S CiA H16 03 (14 H16 04 C14 H16 06 C14 H16 07 CiA C14 CiA H18 H18 H18 N2 N2 0 03 06 52 C14 H18 03 CiA CiA (14 CiA H18 H19 H20 H20 04 N 02 $2 03 N2 04 C14 H20 02 @ C14 H21 CL2 C14 C14 CiA C14 H21 H22 H22 H22 N 03 N 0 N2 02 N2 06 CiA (14 02 CiA H23 H24 N BR2 H24 N 0 N2 N 03+ C14 H24 N2 07 C14 H25 CL3 29491 29496 29876 29338 (14 H16 N2 02 C14 Ci4 29877 FORMULASENTRYP405.(16(16 0629133(16 H16 N6 H16 0229140 29239 29758 2951629515(16 (15 29771 29453 C13 H22 N2 C14 C14 C14 (14 (14 NOS. HBR C13 H19 N 04 C13 H20 CL2 N2 C13 ENTRY (14 C13 (13 H18 04 (13 H19 (L2 N 0 C13 H19 I 08 . FORMULAS 555 29835 29340 28894 29079 29039 29212 28938 29553 29262 29136 C15 (15 (15 (15 . 29892 29430 (15 . H22 H22 H23 H23 CL? 0 BR 02 N 02 CL3 N 03 N2 02 52 04 BR 02 N2 N2 04 5 N4 04 5 0 02 03 N • HCL N 0 N 02 N2 0 N2 S 0 08 52 N 0 N3 0 AR N 02 N+ BR N2 03 N6 02 03 06 N 03 N2 29554 29032 29213 02 04 29537 29924 N2 N2 0 29214 29759 29342 29676 29048 29519 28939 29343 29708 29463 29385 29150 29730 29104 29709 29923 29623 29544 29556 29259 29922 28849 29421 29251 29644 29741 29128 28883 29706 29541 29341 28846 29252 HCLC16 29470 28838 29775 28940 29879 28856 28858 29250 29249 N3 28942 29253 28941 29779 HCL H23 05 HCL 29344 29238 2921S 29028 29237 29243 (16 H9 N 02 S (16 C16 C16 (16 C16 HiO Hil H11 H12 H13 07 F3 02 N 02 N2 02 N3 09 29645 29529 29345 29057 53 H14 CL N 02 Ci6 H14 03 C16 C16 (16 C16 C16 (16 C16 29880 29077 HCL C16 P413 N5 03 C16 H15 HiS H16 H16 H16 H16 H16 0529710(16 H2? 01028857(16 H22 0229093• H23-N HCL(16 0529926(16 H23 N 529442(16 H23 N 06 0829129(16 H24 P44 HCL29217(16 H2S N3 • 029218(16 H2S P43 029348(16 H26 N2 0429568(16 H28 CL29711(16 H31 0229402(16 H32 N2 H32 0229240 2924829242(16 N229403(17(17 H34 29089 •2 HCL . 28847 29834 29526 29422 C16 29056 29760 29485 28884 02 03 N N 02 (15 H28 04 C15 H30 02 C15 H30 03 29260 29514 29080 CiS H26 N2 Cis H26 02 (15 H28 N2 0 29643 29878 294-45 I— 29106 29611 28923 0 S 29339 (15 H1O C1S Hil (15 Hil (15 H12 (15 H12 CiS H12 (15 H13 (15 H14 (15 H14 (15 H14 (15 H14 (iS H14 (15 H14 (15 HiS (15 H15 (15 HiS (15 H16 (15 H16 (15 H16 (15 H16 (15 H17 (15 Hi7 (15 H18 (15 H18 (15 H18 (15 H18 (15 H18 (15 H18 (15 H19 (15 H20 • HBR (15 H20 (15 H20 (15 • HCL (15 H22 C1S H22 0328898C16 H16 02934629733(16 H17 N 0229732(16 H17 N N28943(16 H18 CL N229475(16 H18 029836(16 H18 N4 5229054C16 H18 N4 0929615(16 Hi8 N8 HCL29115(16 Hl9 N • 0429678(16 H20 CL N 0229423(16 H2O HG N22948129495(16 H2O 029347(16 H20 P42 022414139(16 H20 N4 0478854(16 H2O SI29748(16 H20 0429925(16 H21 CL2 N 0229081• H21 P43 HCL(16 0428896. H22 N2 N 0 N7 06 AS N 03 12 04 N2 0 N2 02 N2 04 29902 29677 29761 29216 29881 29165 29528 29401 29464 29646 29247 29560 0229944(17 Hil CL 5329577(17 H12 N2 0 022905829059C17 H13 N S29589(17 Hi'. 03 052941029521(17 H14 0229712(17 H15 CL 0329066(17 HiS 029679(17 H16 BR P43 N28976• H17 CL2 HCL(17 S29713(17 H18 N2 04 029424(17 H18 HCL28944(17 H18 04 • P4,029349(17 H19 029100• Hi9 N HCL(17 N329350(17 Hi9 029882(17 H20 P42 0428945(17 H20 N2 02915729219(17 H20 042885529031(17 H20 029351(17 H21 N 029220. H21 N HCL(17 N329718C17 H21 029833C@7 H21 N3 H22 CL N2 0+ H22 N20229083 28946. HCLCl? 029090• H23 N3 HCL(17 P4529828(17 H23 0229092Ci7 H24 N2 H25 N5 01029937 CancerResearch 556 FORMULAS ENTRY NOS. FORMULASENTRYNOS.C19C19 FORMULASENTRYNOS.C21C21 N228950C19 H22 029178• H23 N HCLC19 028970‘C19 H24 CL N H20 N2 0 C21 H20 OS C21 H20 S C21 H21 AS C17 C17 H32 02 C17 H33 N 02 . 29?44 29174 HBR C17 H34 02 29027 29241 . C18 0228971. H24 CL N HCLC19 C18 H9 AS RR3 N3 (18 C18 C18 C18 C18 Hi0 Hi0 H12 H12 H12 NS 06 AS N2 04 06 S f3R3 02 528922C19 H27 N 02 0229776C19 H28 N2 022923?C19 H28 0229616C20C20 H37 N AS AS 8R2 AS 0? CL P44 02 N4 02 03 28948 29511 28949 29927 29067 29153 29068 BR? 29903 29847 29221 28843 N2 N2 02 P46 0? 0 AS NI AS N3 0 02 07 CL 02 CL 03 NO N2 04 5 P46 07 N 02 N 0+ I— NO 29749 29431 29842 29789 28885 28886 29386 29525 29731 28881 29222 29715 29613 29716 29110 29141 N OS 29680 29510 0? Ci8 H16 Cl8 H16 C18 H16 C18 H16 Cl8 H18 C18 H18 C18 H18 C18 H18 C18 H19 C18 H19 C18 H19 Ci8 H2O C18 H2O Ci8 H2i Ci8 H22 C18 H23 •HCL CiB H?3 Cl8 H24 C18 03+29086C19 H25 N2 28926 28833 06 C18 H13 CiB HiS CiR Sill • H2 0 C18 H13 C18 H14 Ci8 H14 CIA H16 N? 28947 H26 S 06 N2 29780 29570 29180 • HAR C18 H26 N2 02 29087 C18 Ci8 C18 C18 C18 C18 C18 H3O H34 H34 H35 H36 H36 H39 02 04 CL 0 S CL3 04 P 02 04 P 29098 29257 29714 28921 29602 29029 29025 HiO Hi3 H13 Hi3 H13 H13 Hi4 HiS HiS H16 H16 H17 H17 H17 H17 H17 P44 06 AS 8R2 0 AS CL2 0 AS 12 02 AS 03 BR P42 04 02 CL N2 0 N 02 N2 0 OS AS N 0 N 02 P43 08 29883 28887 29173 28888 28889 28824 28890 29750 29352 29751 29647 29146 29353 29648 29354 29465 N? 29790 0 29099 HCLC20 029095‘C2O H30 P42 08794?5C20 H3O N4 H3O 0229234 2923629235C20 0528859C20 H3O 0229224• H31 N HCLC2O 0229245C2O H32 02+29929C2O H33 N2 C19 C19 C19 C19 Ci9 C19 C19 C19 C19 C19 C19 C19 C19 C19 C19 C19 C19 . C19 C19 C19 C19 1/2 H18 H20 H20 H21 BA SALT P42 OS 06 N 04 5 29387 29524 29523 29441 CL42981953R4 H6 04C20 N429359C20 H1O 0429818C20 H13 CL 0429156C2O H13 I I29151C?0 Hi4 AS 042984029841C20 H14 NB 529846• H14 N8 07 SALTC20 NA 0229626C20 H14 0329762C20 H14 029763C20 HiS N 5329578C20 H16 N2 0 S28825C2O H16 N2 04 0229764C20 H16 5228908C20 H16 02 CL28891C2O H17 0429884C?0 H20 P42 0228826C2O H22 BR N CL229681N2 H22 04C20 OS29989C2O H22 NB 0328877C2O H22 0229404C20 H24 N2 0229928C20 H24 0229223C20 H2S N 0229781• H25 N HCLC20 028975• H26 CL N HCLC2O 0229765C2O H26 N 0229824C2O H26 N4 0229766C2O H27 N 0228829. H27 N 029930C2O H37 N 0429571C20 H37 N 5228903C20 H38 0429246C20 H4O 0229125C2O H41 N N29618C21C21 H43 N29388C21 HiS 0429848C21 H16 P48 028892C21 H16 0329650C21 H17 N S29052C21 H17 N 01? 0229049C21 Hi7 N3 Hi8 0228830 HG C21 H23 N 03 C21 H24 N2 S C21 H24 09 C21 H27 N7 014 P2 C21 H32 N4 08 C21 H32 02 C21 H39 N 0 C21 H41 N 02 C21 H43 N 0329405 29885C22C22 HiS AS 28831 29813 29522 29993 29426 29233 29931 29617 S C22 HiS CL4 N 04 C2? Hi8 03 C22 H19 N C27 H19 N 04 C22 H2? N2 0 C22 H23 CL N 08 •SB(I1I) CL3 DERIV. 2418?'3 2895? 29427 29817 29358 2993? C22 29933 . H24 N 08 SR(I11) CL3 DFR!V. C22 H24 P44 •2 HCL C2? H2S N3 0 • HCL C22 H26 P44 06 52 C?? H79 N 0 . . 29091 29088 29435 29226 HCL C22 H29 N 02 29782 HCL C22 H30 CL N 0 • HCL C27 H3O P42 •2 HCL 28972 28953 2965229934C23C?3 C22 H42 N? 029169 H17 AS C23 H18 29627 C23 H18 0 29158 C23 H22 03 28832 C23 H24 CL? N2 29794 C23 H25 CL N2 0 29810 C23 H25 N3 29355 C23 H25 N3 02 29802 C23 H26 N2 0 29811 C23 H26 N2 03 S 29795 • NA SALT C23 H30 N2 29820 C23 H38 CL N 028893 29620C24C24 02 C24 C24 C24 C24 . 29649 CL 29520 29225 29138 C24 C24 C24 C24 C24 . HiS 53 H16 H17 H17 H19 CL2 H2O H21 H22 H23 H24 CL N2 29579 N8 04 AS N AS 29845 29070 29147 29071 HG 04 N3 AS2 N2 0 N CL N 0 HCL C24 H2S N 0 C24 28954 28955 29172 29486 28974 H26 AS+ 29472 CL 29177 29651 Index of Materials FORMULAS ENTRY NOS. 557 ENTRY FORMULAS P405. C24 C36 C24 H26 P42 02 C24 H26 P42 02 • NA SALT 29799 29805 C24 29797 29793 29806 H28 P42 C24 H28 P42 02 C24 H28 P42 04 S . NA 29826 C36 H27 • 8R2 MG 29176 C36 H27 AS C36 H34 02 29734 C36 H72ASN2S 0429142 29132C37C37 SALT C24 H30 N2 02 C24 H37 N 02 C24 H42 29102 29935 28834 HS4020229469 29767C38C38H76N2OS29612C39C39H42P4229809C40C4OH46P4429814C42C42 C37H52 C25 N 015 S2 29051 AS 0+ I— 29152 CL P42 29798 29796 P43 0 N2 02 29791 29800 C2S H30 07 29530 C25 H32 04 29527 C2S C2S C2S C2S C2S H18 H22 H25 H29 H30 29792 29807 C26 C26 H18 C26 H18 05 C26 H19 AS 0 . H2 C4 H4 P42 06 S 04 F 07 P49 09 53 SALT 04 p P42 P42 29654 29655 29784 29055 29886 29803 29097 04 C27 C27 C27 C27 C?7 H20 H28 HIS H35 P42 07 P42 0 P43 P43 02 29155 29812 29804 29801 C28 H2O P42 H28 AS2 N2 29227 29073 H28 A52 OS H30 P42 03 H31 P42 03+ 29171 29821 28969 H34 015 H42 02 29936 28835 C29 H28 012 54 C29 H37 CL? NI 29583 29808 C28 C28 03 C28 C28 C28 CL C28 C28 52 H72N4N206 C42H46 0 C26 H20 C26 H2O C26 H21 C26 H29 •3 NA C26 H31 C26 H32 C26 H36 . 29581 29653 29072 C29 C30 C30 H30 P44 04 S C30 H32 P42 28836 28956 C32 C32 H14 P48 012 C32 H28 P42 C32 H28 P42 04 29887 28957 29074 C34 C34 H14 BR8 08 C34 H18 010 C34 H22 08 29816 29822 29815 29785 29135 29619 2975? INORGAN IC COMPOUNDS CA CL CL H2 H4 04 P2 K 04 NA 03 NA 02 P H3 02 28978 28979 28987 28984 p 29010 NA2S •9H2O P4A2 54 28980 28985 MATERIALS FORMULAS SULFONATED SALT UREASE WITHOUT SPAN 80, SODIUM 29446 29893 NOTES NOTES NOTES INSTRUCTIONS FOR AUTHORS ON THE PREPARATION OF DATA FOR SUPPLEMENTS Data submitted for publication in the supplements on “CancerChemotherapy Screen-. ing Data― should be sent to Dr. Joseph Leiter, National Cancer Institute, Bethesda 14, Maryland. Deadline.,.—Thedeadlines for the receipt of papers are February 1, June 1, and October 1 of each year; the supplements will appear about four months later. 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Each paper should include a brief but specific section on Materials and Methods, in eluding such information as how the compounds were administered, what solvents were used, what dose schedules were followed, the source of the compounds, diet of the animals, etc. In particular, the authors should indicate the basis upon which they judge the sig nificance of their finding. Any abbreviations used should be clearly defined in footnotes. The tables should follow the general style of the present supplement, should be supplied with an appropriate Since the major objective presentation of tabular data, a résumé of the significant When used, references of these supplements summaries, and every column heading. is to provide a medium when included, should for adequate be brief and restricted to results presented. to the literature should be listed according to the style used in Cancer Research, One hundred authors, reprints of each article, if desired, will be furnished without charge to A
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